| Cat.No.: | BSM-0352 |
| Product Name: | Cyproheptadine (hydrochloride hydrate) |
| CAS No.: | 41354-29-4 |
| Figure: |
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| Product Overview: | A first-generation antihistamine |
| Description: | Cyproheptadine is a first-generation antihistamine that potently antagonizes the histamine H1 receptor (pKi = 9.42). It also antagonizes serotonin and muscarinic receptors at nanomolar concentrations. Cyproheptadine also inhibits the lysine methyltransferase SET7/9 (IC50 = 1 µM), suppressing the expression of estrogen receptor α in human breast cancer MCF-7 cells. |
| Appearance: | A crystalline solid |
| Molecular Weight: | 350.9 |
| Purity: | ≥98% |
| Storage: | -20°C |
| Targets: | Lysine methyltransferase SET7/9 |
| Molecular Formula: | C21H21N • HCl [1.5H2O] |
| Chemical Name: | 4-(5H-dibenzo[a,d]cyclohepten-5-ylidene)-1-methyl-piperidine, monohydrochloride, sesquihydrate |
| Warning: | For Research Use Only! Not For Use in Humans. |
| Product Types | ||
| ◆ Bioactive Small Molecules | ||
| BSM-0027 | UNC0321 (trifluoroacetate salt) | Inquiry |
| ◆ Antibodies | ||
| EAb-0030 | SETD8 Polyclonal Antibody | Inquiry |
| EAb-0031 | SETDB1 Polyclonal Antibody | Inquiry |
| EAb-0032 | Setd1a Polyclonal Antibody | Inquiry |
| EAb-0033 | Setd1b Polyclonal Antibody | Inquiry |
| Related Gene / Proteins | |||
| SENP3 | SENP8 | SET | SET1 |
| SET2 | SET7 | SET8 | SET9 |
| SETBP1 | SETD1A | SETD1B | SETD2 |
| SETD3 | SETD5 | SETD6 | SETD7 |
| SETD8 | SETD9 | SetDB1 | SETDB2 More > |
| SETMAR | |||
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