Cat.No.: | BSM-0343 |
Product Name: | MS023 (hydrochloride) |
CAS No.: | 2108631-19-0 |
Figure: | |
Product Overview: | An inhibitor of type I PRMTs |
Description: | MS023 is a potent, selective inhibitor of type I PRMTs (IC50s = 20, 119, 83, 8, and 8 nM for PRMT1, 3, 4, 6, and 8, respectively). It is inactive against type II and type III PRMTs, as well as other types of MTs. MS023 is active in cells, inhibiting the dimethylation of histone 4 at Arg3 by PRMT1 with an IC50 value of 9 nM. |
Appearance: | A crystalline solid |
Molecular Weight: | 396.8 |
Purity: | ≥95% |
Storage: | -20°C |
Targets: | type I PRMTs |
Molecular Formula: | C17H25N3O • 3HCl |
Chemical Name: | N1-methyl-N1-[[4-[4-(1-methylethoxy)phenyl]-1H-pyrrol-3-yl]methyl]-1,2-ethanediamine, trihydrochloride |
Warning: | For Research Use Only! Not For Use in Humans. |
Product Types | ||
◆ Bioactive Small Molecules | ||
BSM-0027 | UNC0321 (trifluoroacetate salt) | Inquiry |
BSM-0047 | SGC707 | Inquiry |
◆ Antibodies | ||
EAb-0048 | PRMT6 Polyclonal Antibody | Inquiry |
EAb-0049 | PRMT7 Polyclonal Antibody | Inquiry |
EAb-0050 | PRMT1 Polyclonal Antibody | Inquiry |
Related Gene / Proteins | |||
Pr-SET7 | PRC1 | PRC2 | PRDM1 |
PRDM10 | PRDM11 | PRDM12 | PRDM13 |
PRDM14 | PRDM15 | PRDM16 | PRDM17 |
PRDM2 | PRDM3 | PRDM4 | PRDM5 |
PRDM6 | PRDM7 | PRDM8 | PRDM9 More > |
PREP1 | PRIM2 | PRKAA2 | PRKCA |
PRKCB | PRKCE | PRKDC | PRKRIP1 |
PRMT | prmt1 | PRMT2 | PRMT3 |
PRMT5 | prmt6 | PRMT7 | PRMT8 |
PRMT9 | Progerin | Protamine 2 | Prox1 |
PRPF31 | PRPF40A | PRSS12 | PRSS55 |
PRTFDC1 |
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