| Cat.No.: | BSM-0195 |
| Product Name: | PFI-4 |
| CAS No.: | 900305-37-5 |
| Figure: |
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| Synonyms: | N-[2,3-Dihydro-1,3-dimethyl-2-oxo-6-(1-pyrrolidinyl)-1H-benzimidazol-5-yl]-2-methoxybenzamide |
| Description: | PFI-4 is a potent and selective BRPF1 bromodomain inhibitor (IC50 = 80 nM). Displays >100-fold selectivity for BRPF1 over a panel of other bromodomains including BRPF2 (BRD1), BRPF3 and BRD4. |
| Appearance: | Pale green solid |
| Molecular Weight: | 380.44 |
| Purity: | ≥ by HPLC |
| Storage: | -20°C |
| Targets: | BRPF1 bromodomain |
| Molecular Formula: | C₂₁H₂₄N₄O₃ |
| MDL Number: | N/A |
| Solubility: | >15 mg/ml (DMSO) |
| Shipping Conditions: | Gel Pack |
| Warning: | For Research Use Only! Not For Use in Humans. |
| Product Types | ||
| ◆ Synthetic Peptides | ||
| SP-0001 | Bromodomain Non-Acetylated Ligand 4 | Inquiry |
| SP-0002 | Bromodomain Non-Acetylated Ligand 3 | Inquiry |
| SP-0003 | Bromodomain Non-Acetylated Ligand 1 | Inquiry |
| SP-0004 | Bromodomain Ligand 3 | Inquiry |
| SP-0006 | Bromodomain Ligand 4 | Inquiry |
| Related Gene / Proteins | |||
| BRCA1 | BRCA2 | BRCC3 | BRD |
| brd1 | brd2 | brd3 | brd4 |
| BRD7 | BRD8 | brd9 | brdt |
| BRL | BRM | BRMS1 | BRPF1 |
| BRPF2 | brpf3 | BRWD1 | BRWD3 |
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