| Cat.No.: | BSM-0169 |
| Product Name: | Mocetinostat (MGCD0103) |
| CAS No.: | 726169-73-9 |
| Figure: |
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| Synonyms: | N-(2-Aminophenyl)-4-[[[4-(3-pyridinyl)-2-pyrimidinyl]amino]methyl]benzamide; Mocetinostat; MG0103 |
| Description: | Mocetinostat (MGCD0103) selectively inhibits histone deacetylases (HDACs) 1-3 and 11 at submicromolar concentrations. (IC50 = 0.15, 0.29, 1.66 and 0.59 µM for HDAC1, 2, 3 and 11 respectively). Mocetinostat induces hyperacetylation of histones, causes expression of the tumor suppressor protein p21(WAF1/CIP1), and inhibits proliferation of human cancer cells growing in culture. |
| Appearance: | White to off-white solid |
| Molecular Weight: | 396.44 |
| Purity: | >98% by HPLC |
| Storage: | -20 ̊C |
| Targets: | Class I HDAC |
| Molecular Formula: | C23H20N6O |
| MDL Number: | MFCD03453554 |
| Solubility: | DMSO |
| Shipping Conditions: | Gel Pack |
| Warning: | For Research Use Only! Not For Use in Humans. |
| Product Types | ||
| ◆ Extracts & Lysates | ||
| EL-0006 | Recombinant Human HDAC1 293 Cell Lysate | Inquiry |
| EL-0007 | Recombinant Human HDAC2 293 Cell Lysate | Inquiry |
| EL-0008 | Recombinant Human HDAC3 Cell Lysate | Inquiry |
| EL-0009 | Recombinant Human HDAC4 Cell Lysate | Inquiry |
| ◆ Bioactive Small Molecules | ||
| BSM-0007 | Tubacin | Inquiry |
| Related Gene / Proteins | |||
| HDAC | HDAC1 | HDAC10 | HDAC11 |
| HDAC2 | HDAC3 | hdac4 | hdac5 |
| HDAC6 | hdac7 | HDAC8 | hdac9 |
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