Cat.No.: | BSM-0168 |
Product Name: | ME-0328 |
CAS No.: | 1445251-22-8 |
Figure: |
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Synonyms: | 3,4-Dihydro-4-oxo-3,4-Dihydro-4-oxo-N-[(1S)-1-phenylethyl]-2-quinazolinepropanamide |
Description: | ME-0328 is a potent and selective PARP-3 inhibitor (IC₅₀ = 0.89 µM). ME-0328 inhibits PARP-1, PARP-2 and other ARDTs (ADP ribosyltransferases) at much higher concentrations (IC₅₀ = 6.3, 10.8 and >30 µM, respectively). |
Appearance: | White solid |
Molecular Weight: | 321.37 |
Purity: | ≥98% by TLC |
Storage: | -20°C |
Targets: | PARP-3 |
Molecular Formula: | C₁₉H₁₉N₃O₂ |
MDL Number: | MFCD03453554 |
Solubility: | DMSO (~30 mg/ml) or EtOH (~4 mg/ml) |
Shipping Conditions: | Gel Pack |
Warning: | For Research Use Only! Not For Use in Humans. |
Product Types | ||
◆ Antibodies | ||
EAb-0059 | PARP Monoclonal Antibody | Inquiry |
EAb-0061 | PARP Polyclonal Antibody | Inquiry |
EAb-0062 | PARP (Cleaved) Polyclonal Antibody | Inquiry |
EAb-0063 | PARP (Cleaved) Polyclonal Antibody | Inquiry |
EAb-0064 | Paf1 Polyclonal Antibody | Inquiry |
Related Gene / Proteins | |||
PABPC1L2A | PABPC5 | PABPN1 | PAD |
PAD1 | PAD2 | PAD3 | PAD4 |
PADI1 | PADI2 | PADI3 | PADI4 |
PADI6 | PAF1 | PAN2 | PAPD1 |
PAPD4 | PAPD5 | PAPD7 | PAPOLA More > |
PAPOLB | PARD6A | PARG | PARK2 |
PARK7 | PARP | PARP1 | PARP10 |
PARP11 | PARP12 | PARP14 | PARP15 |
PARP16 | PARP2 | PARP3 | PARP4 |
PARP6 | PARP7 | PARP8 | PARP9 |
PAX5 | PAX6 | PAX7 | PAX9 |
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