Cat.No.: | BSM-0030 |
Product Name: | PF-06405761 |
CAS No.: | 1403764-72-6 |
Abbr: | PF-06405761(BRD4) |
Synonyms: | CAP, HUNK1, HUNKI, MCAP |
Description: | PF-06405761 is a selective BET (bromodomain-containing protein) inhibitor for BRD4 with IC50 of 0.22 μM. |
Molecular Weight: | 347.39 |
Purity: | > 95% |
Storage: | 4°C |
Targets: | BRD4 |
IC50: | 0.22 μM |
Molecular Formula: | C16H17N3O4S |
Chemical Name: | 2-methoxy-N-(3-methyl-2-oxo-1,2,3,4-tetrahydroquinazolin-6-yl)benzenesulfonamide |
Warning: | For Research Use Only! Not For Use in Humans. |
Product Types | ||
◆ Synthetic Peptides | ||
SP-0001 | Bromodomain Non-Acetylated Ligand 4 | Inquiry |
SP-0002 | Bromodomain Non-Acetylated Ligand 3 | Inquiry |
SP-0003 | Bromodomain Non-Acetylated Ligand 1 | Inquiry |
SP-0004 | Bromodomain Ligand 3 | Inquiry |
SP-0006 | Bromodomain Ligand 4 | Inquiry |
Related Gene / Proteins | |||
BRCA1 | BRCA2 | BRCC3 | BRD |
brd1 | brd2 | brd3 | brd4 |
BRD7 | BRD8 | brd9 | brdt |
BRL | BRM | BRMS1 | BRPF1 |
BRPF2 | brpf3 | BRWD1 | BRWD3 |
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